Carbetapentane Citrate CAS 23142-01-0

What is Carbetapentane Citrate CAS 23142-01-0?

Carbetapentane Citrate CAS 23142-01-0, also known as pentoxyverine citrate, is a pharmaceutical intermediate and research compound functioning primarily as an antitussive (cough suppressant) and sigma-1 receptor agonist. It appears as a white to off-white solid and is typically used in biochemical studies and preclinical models exploring respiratory mechanisms, central nervous system modulation of the cough reflex, and related pharmacological pathways.

Specification

Feature

• Antitussive Pharmacological Activity: CARBETAPENTANE CITRATE is recognized for its cough-suppressing activity, working through central modulation of the cough reflex, making it relevant in respiratory pharmacology research models.
• Sigma-1 Receptor Agonist: Acts as a ligand at the sigma-1 receptor, a target implicated in neurological signal modulation, offering utility in neuropharmacology and receptor research.
• Water-Soluble Citrate Salt: The citrate form enhances solubility compared with the parent compound, facilitating formulation in aqueous systems for analytical and experimental use.
• Research Reference Standard: Due to its well-defined pharmacological profile, CARBETAPENTANE CITRATE is used as a reference compound in HPLC/LC-MS and other analytical assays in pharmaceutical R&D settings.

Application

• Respiratory Pharmacology Research: Used in in vitro and preclinical studies to investigate mechanisms of cough suppression, airway responsiveness, and central nervous system control of respiratory reflexes.
• Sigma-1 Receptor Studies: Employed in biochemical and cell signaling research focused on sigma-1 receptor function and modulation.
• Drug Discovery & Screening: Applied as a screening compound in early-stage pharmaceutical research evaluating antitussive and CNS-active candidates.
• Analytical & Reference Uses: Used as a reference standard or analytical intermediate in method development for respiratory drug analysis.

Packaging

Mikem offers flexible packaging options, including 25 kg of fiber drums for liquid products and 15–25 kg PP/PE bags for powder products, all customizable to meet your specific needs.